Melanotana 1he tairitenga peptide waihanga oα-MSH (alpha-melanocyte stimulating hormone). Ka mahi nate whakahohe i nga kaiwhakawhiwhi melanocortin-1 (MC1R)ki te whakaongaongahanga melanin, tuku maorikiri kiriawhakamarumaru whakaahua.
Kua otikua whakaaetia mo te maimoatanga o te erythropoietic protoporphyria (EPP)—he mate onge e pa ana ki te ra. Ka awhina a Melanotan 1 ki te piki akete manawanui ki te rama UV, whakaititauhohenga phototoxic, me te whakarei akete tiaki kiri ki te kino o te UV.
WhiriwhiriMC1R agonist
Ka piki akehanga eumelanin
Ka whakaratotiaki ra maori
TautokoTe whakatikatika DNA me te whakautu anti-inflammatory
Pmanawanui movitiligo, ārai mate pukupuku kiri, apigmentation whakapaipai
I tirotirohia ki rotoanti-pakekeamaimoatanga dermatological
Te parakore teitei ≥99%
Te whakahiato peptide-waa totoka (SPPS)
Nga paerewa hangahanga rite-GMP
Te tuku tauine: R&D ki nga taumata arumoni