Melanotana IIhe tairitenga heptapeptide hurihanga waihanga oα-melanocyte-stimulating hormone (α-MSH), whakawhanakehia kiwhakaongaonga i te melanogenesis, whakareiTiaki UV, me te whakarerekemahi moepuku me te metabolic. Ka mahi hei aagonist kore-whiriwhirio nga kaiwhakawhiwhi melanocortin, ina koaMC1R, MC3R, aMC4R.
I ako tuatahi mo onatanningatiaki whakaahuataonga, kua whakaatu hoki a Melanotan II nga paanga ki rungate whakanui i te libido, te whakakore i te hiahia, ataurite pūngao, ka waiho hei peptide rangahau multifunctional me te hiahia ki te dermatology, endocrinology, me te rongoa moepuku.
Ka mahi a Melanotan II ma te whakahohe i te maha o nga kaiwhakawhiwhi melanocortin:
MC1R: Whakatairangahanga melanin→ whakanui ake i te kiri kiri me te whakamarumaru UV
MC3R / MC4R: Kua uru ki rotowhakahaere hiahia, te whakanui i te libido, ahomeostasis pūngao
Ka whakawhiti i te arai toto-roro, te awe i nga huarahi neurohormonal pokapū
Ahakoa kaore i whakaaetia mo te whakamahi rongoa, ka akohia a Melanotan II mo nga mea e whai ake nei:
Whakatairangate whakahiato eumelanin, ka arahi kitanning maori
Ka whakaratopānga tiaki whakaahuame te kore e pa ki te ra
He kaha mo te whakaheke i te mate pukupuku kiri i roto i nga tangata kiri-tika
Ka whakaatuhia kite whakanui i te libido me te whakaihiihii roto i nga tane me nga wahine
I ako hei rongoa momate erectile (ED)mā te whakahohenga MC4R
Meiwhakaitihia te hiahia me te kai kaima te mahi i runga i nga huarahi hypothalamic
He taapiri pea ki rotorangahau mōmona
Te parakore teitei ≥ 99%(HPLC & LC-MS kua whakapumautia)
I whakahiato mate whakahiato peptide-waa toka (SPPS)
He iti te endotoxin, he iti te toenga whakarewa
Kei te waatea i rotoR&D ki te tauine arumoni