Pharma APIs
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Fmoc-His-Aib-OH
Ko te Fmoc-His-Aib-OH he poraka hangahanga dipeptide e whakamahia ana i roto i te whakahiato peptide, te whakakotahi i te histidine kua tiakina e Fmoc me te Aib (a-aminoisobutyric acid). Ka whakaatu a Aib i te rigidity conformational, he mea nui mo te hoahoa peptides helical me te pumau.
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Boc-Tana(Trt)-Aib-Glu(OtBu)-Gly-OH
Ko te Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH he kongakonga tetrapeptide kua tiakina e whakamahia ana i roto i te whakahiato peptide me te whanaketanga tarukino. Kei roto i nga roopu mahi kua parea rautaki mo te hono takahanga me te whakaatu i te Aib (a-aminoisobutyric acid) hei whakarei ake i te pumau o te helix me te rigidity conformational.
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Ste-γ-Glu-AEEA-AEEA-OSU
Ko te Ste-γ-Glu-AEEA-AEEA-OSU he ngota ngota whakahiato lipid kua hangaia mo te tuku raau taero me te whakakotahi i nga raau taero antibody (ADC). Kei roto i te stearoyl (Ste) hydrophobic hiku, he γ-glutamyl motif arotahi, AEEA mokowhiti mo te ngawari, me te roopu OSu (NHS ester) mo te whakakotahi pai.
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Fmoc-Ile-αMeLeu-Leu-OH
Ko te Fmoc-Ile-αMeLeu-Leu-OH he paraka hanga tripeptide kua parea ki te waihanga e whakaatu ana i te α-methylated leucine, e whakamahia nuitia ana i roto i te hoahoa tarukino peptide hei whakarei ake i te pumau o te tinana me te kowhiringa o te kaikawe.
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Dodecyl Phosphocholine (DPC)
Ko te Dodecyl Phosphocholine (DPC) he waipara zwitterionic waihanga e whakamahia nuitia ana i roto i te rangahau pūmua membrane me te koiora hanganga, ina koa i roto i te NMR spectroscopy me te crystallography.
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Ko te Caspofungin mo nga Infections Antifungal
Ingoa: Caspofungin
Nama CAS: 162808-62-0
tātai rāpoi: C52H88N10O15
Te taumaha ngota: 1093.31
Nama EINECS: 1806241-263-5
Ira kohua: 1408.1±65.0 °C (Te Matapae)
Kiato: 1.36±0.1 g/cm3(Whakaahua)
Te whakarea kawatanga: (pKa) 9.86±0.26 (Te Matapae)
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Daptomycin 103060-53-3 mo nga mate hopuhopu
Ingoa: Daptomycin
Nama CAS: 103060-53-3
tātai rāpoi: C72H101N17O26
Te taumaha ngota: 1620.67
Tau EINECS: 600-389-2
Ira whakarewa: 202-204°C
Ira kohua: 2078.2±65.0 °C (Te Matapae)
Kiato: 1.45±0.1 g/cm3(Whakaahua)
Ira hiko: 87℃
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Micafungin mo te antifungal me te antiviral
Ingoa: Micafungin
Nama CAS: 235114-32-6
tātai rāpoi: C56H71N9O23S
Te taumaha ngota: 1270.28
Nama EINECS: 1806241-263-5
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Ko te Vancomycin he paturopi glycopeptide e whakamahia ana mo te paturopi
Ingoa: Vancomycin
Te nama CAS: 1404-90-6
tātai rāpoi: C66H75Cl2N9O24
Te taumaha ngota: 1449.25
Tau EINECS: 215-772-6
Kiato: 1.2882 (whakatau tata)
Taupū Reractive: 1.7350 (whakatau tata)
Nga tikanga rokiroki: hiri ki te maroke, 2-8°C
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Ko te Vardenafil Dihydrochloride e rongoa ana i te mate erectile 224785-91-5
Nama CAS: 224785-91-5
tātai rāpoi: C23H32N6O4S
Te taumaha ngota: 488.6
Tau EINECS: 607-088-5
Ira whakarewa: 230-235°C
Kiato: 1.37
Irahiko: 9℃
Nga tikanga rokiroki: Kua hiri ki te maroke, Rokiroki ki te pouaka tio, i raro i te -20°C
Te whakarea kawatanga: (pKa) 9.86±0.20 (Whakaahua)
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Orlistat 96829-58-2 Te whakaiti i te whakauru o te ngako Sietary, ka hua ki te mate taimaha
Nama CAS: 96829-58-2
tātai rāpoi: C29H53NO5
Te taumaha ngota: 495.73
Tau EINECS: 639-755-1
Te hurihanga motuhake: D20-32.0°(c=1inchloroform)
Ira kohua: 615.9±30.0°C (Whakaahua)
Kiato: 0.976±0.06g/cm3(Whakaahua)
Nga tikanga rokiroki: 2-8°C
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Ko te RU-58841 i whakamahia hei aukati i nga makawe me te pakira tauira tane
CBN nama:CB51396657
Ingoa:RU 58841
Nama CAS: 154992-24-2
tātai rāpoi: C17H18F3N3O3
Te taumaha ngota: 369.34
Nama EINECS: 1592732-453-0
