Hexarelinhe waihangapeptide secretagogue hormone tupu (GHS)me te kahaGHSR-1a agonist, i whakawhanakehia hei whakaongaongatukunga homone tupu endogenous (GH).. No tewhanau ghrelin mimetice ono nga waikawa amino (he hexapeptide), he pai ake te whakapumautanga o te metabolic me te kaha ake o te tuku GH ki nga tairitenga o mua penei i te GHRP-6.
Hexarelin te ako whanui mo ona tono i roto ite endocrinology, te whakamarumaru o nga uaua, te whakatikatika ngakau, me nga maimoatanga aukati i te koroheketanga, na tona kaha ki te whakanui i te GH me teTauwehe tipu rite-insulin 1 (IGF-1)nga taumata kaore i te whakauru tika i nga homoni o waho.
Hexarelin here ki tekaikawe huna huna homone tupu (GHSR-1a)i runga i te pituitary me te hypothalamus, e pee ana i te mahi akerelin—te hiakai maori o te tinana me te homoni tuku GH.
Nga mahi ahuwhenua matua:
Ka whakaihiihi i te tukunga GH pulsatile
Ka piki te hurihangaIGF-1taumata
Whakatairangapānga anabolic(te tipu o te uaua, te whakaora)
Tautokopākia ngakoawhakahounga pūtau
Ka whakaatu peacardioprotectiveaanti-apoptoticpānga
Kaore i rite ki etahi atu peptides GHS, he mahi a Hexareline kore e tino whakanuia cortisol prolactin ranei, e tuku ana i te tohu endocrine pokekore.
Whakatairangapapatipu tinana hirokiwhanaketanga
Whakarei akete whakatikatika me te whakahou i nga uaua
I ako i rotosarcopenia, cachexia, me te whakaora i muri i te pokanga
Ko nga rangahau preclinical e whakaatu anapai ake te mahi ngakaui muri i te whara myocardial
Ka whakaitifibrosis ngakaume te whakarei akete hautau ejection ventricular maui
Te whakamahi pea i rotongoikore o te ngakauate koroheketanga ngakautauira
Ka piki akelipolysisme te whakapai akete tairongo o te insulin
Tautokorongoā anti-pakekena roto i te whakaongaonga tuaka GH/IGF-1
Ka awhina pea ki te pupurikiato wheua me te hauora tahi
Pure ≥ 99%
I hangaia mate whakahiato peptide-waa toka (SPPS)
Nga paerewa rite GMP, iti te endotoxin me nga toenga whakarewa
Tukunga ngawari:R&D ki te tauine arumoni