Hua
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High Purity Peptides Retatrutide 10mg mo te mate taimaha me te mate huka
Maamaa: >99%
State: Paura Lyophilized
Te ahua: Te paura ma
Whakatakotoranga: 5mg/10mg/15mg/20mg/30mg
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Retatrutide
Ko te Retaglutide he rongoa hou mo te dipeptidyl peptidase-4 (DPP-4) hei aukati i te paheketanga o te glucagon-like peptide-1 (GLP-1) me te polypeptide tuku-insulin-whakaeke (GIP) na te DPP-4 enzyme i roto i te whekau me te toto, ka whakaroa i a raatau mahi, me te kore e pa ki te hangai o te insulin i te wa e pa ana ki te taumata o te insulin. te whakaheke i te hunanga o te glucagon e nga pūtau α pancreatic, na reira ka pai ake te whakahaere i te huka toto postprandial. He pai te mahi i runga i te paanga hypoglycemic, te manawanui, me te tautukunga.
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konutai Inclisiran
Ko te Inclisiran sodium API (Active Pharmaceutical Ingredient) e tino akohia ana i roto i te mara o te wawaotanga RNA (RNAi) me nga rongoa cardiovascular. I te mea he siRNA paerua-rua e aro ana ki te ira PCSK9, ka whakamahia i roto i te rangahau haumanu me te rangahau haumanu ki te arotake i nga rautaki whakaheke ira-a-roa mo te whakaheke i te LDL-C (te cholesterol iti-density lipoprotein cholesterol). Ka noho ano hei tauira tauira mo te tirotiro i nga punaha tuku siRNA, te pumau, me nga rongoa RNA e whaaia ana e te ate.
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Fmoc-Gly-Gly-OH
Ko te Fmoc-Gly-Gly-OH he dipeptide e whakamahia ana hei poraka hanga taketake i roto i te whakahiato peptide-waahanga totoka (SPPS). E rua nga toenga glycine me tetahi N-terminus tiaki-Fmoc, e taea ai te whakaroa o nga mekameka peptide. Na te iti o te rahi me te ngawari o te glycine, ka akohia tenei dipeptide i roto i te horopaki o te hihiri o te tuara peptide, te hoahoa hono, me te whakatauira hanganga i roto i nga peptides me nga pūmua.
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Fmoc-Thr(tBu)-Phe-OH
Ko te Fmoc-Thr(tBu)-Phe-OH he poraka hanga dipeptide e whakamahia nuitia ana i roto i te whakahiato peptide-waahanga totoka (SPPS). Ko te roopu Fmoc (9-fluorenylmethyloxycarbonyl) e tiaki ana i te N-terminus, ko te roopu tBu (tert-butyl) e tiaki ana i te mekameka taha hydroxyl o te threonine. Ka rangahaua tenei dipeptide whakamarumaru mo tana mahi ki te whakahaere i te whakaroa peptide pai, te whakaheke i te raemi, me te whakatauira i nga kaupapa raupapa motuhake i roto i te hanganga pūmua me nga rangahau taunekeneke.
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AEEA-AEEA
Ko te AEEA-AEEA he hauwai, he mokowhiti ngawari e whakamahia nuitia ana i roto i te peptide me te rangahau whakakotahitanga tarukino. E rua nga waeine ethylene glycol, e whai hua ana mo te ako i nga paanga o te roa o te hono me te ngawari ki nga tauwhitinga ngota, te whakarewatanga me te mahi koiora. He maha nga wa ka whakamahia e nga Kairangahau nga waeine AEEA ki te arotake i te awe o nga mokowhiti i te mahi o nga whakangao antibody-drug conjugates (ADCs), peptide-drug conjugates, me etahi atu bioconjugates.
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Fmoc-L-Lys[Eic(OtBu)-γ-Glu(OtBu)-AEEA]-OH
Ko tenei pūhui he parenga, he lysine derivative kua whakamahia i roto i te whakahiato peptide me te whanaketanga conjugate tarukino. Kei roto i te roopu Fmoc mo te whakamarumaru N-terminal, me te whakarereke-taha me te Eic(OtBu) (waikawa heicosanoic derivative), waikawa γ-glutamic (γ-Glu), me te AEEA (aminoethoxyethoxyacetate). I hangaia enei waahanga ki te ako i nga paanga lipidation, te matū mokowhiti, me te tuku raau taero. Kei te rangahau whanui i roto i te horopaki o nga rautaki prodrug, hononga ADC, me nga peptides tauwhitiwhiti membrane.
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Fmoc-L-Lys[Ste(OtBu)-γ-Glu-(OtBu)-AEEA-AEEA]-OH
He pärönaki lysine kua whakarerekëtia te pühui nei e whakamahia ana i roto i te whakahiato peptide, ina koa mo te hanga i nga hononga peptide i whäia, maha-maha ranei. Ka taea e te roopu Fmoc te whakahiato hikoi ma te Fmoc toka-waahanga peptide synthesis (SPPS). Ka whakarereketia te mekameka taha ki te waikawa stearic waikawa (Ste), te waikawa γ-glutamic (γ-Glu), me nga hononga AEEA e rua (aminoethoxyethoxyacetate), e whakarato ana i te hydrophobicity, nga taonga utu, me te mokowhiti ngawari. Kei te rangahauhia mo tana mahi i roto i nga punaha tuku tarukino, tae atu ki nga antibody-drug conjugates (ADCs) me nga peptides-roto-a-roto.
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Liraglutide Anti-Diabetics mo te Mana Huka Toto CAS NO.204656-20-2
Ingredient Active:Ko te Liraglutide (he rite ki te glucagon-like peptide-1 (GLP-1) te tangata i hangaia e te rewena na roto i te hangarau whakakotahitanga ira).
Ingoa matū:Arg34Lys26-(N-ε-(γ-Glu(N-α-hexadecanoyl)))-GLP-1[7-37]
Ētahi atu Kai:Disodium Hydrogen Phosphate Dihydrate, Propylene Glycol, Hydrochloric Acid and/ranei Sodium Hydroxide (hei Whakariterite pH Anake), Phenol, me te Wai mo te Werohanga.
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Ko te Leuprorelin Acetate te whakahaere i te hunanga o nga Hormone Gonadal
Ingoa: Leuprorelin
Nama CAS: 53714-56-0
tātai rāpoi: C59H84N16O12
Te taumaha ngota: 1209.4
Tau EINECS: 633-395-9
Te hurihanga motuhake: D25 -31.7° (c = 1 i roto i te 1% waikawa ahetiki)
Kiato: 1.44±0.1 g/cm3(Whakaahua)
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Boc-Tana(Trt)-Aib-Gln(Trt)-Gly-OH
Boc-Tana(Trt)-Aib-Gln(Trt)-Gly-OHhe tetrapeptide parea e whakamahia ana i roto i te whakahiato peptide me nga rangahau hanganga. Ko te roopu Boc (tert-butyloxycarbonyl) e tiaki ana i te N-terminus, ko nga roopu Trt (trityl) te tiaki i nga mekameka taha o te histidine me te glutamine hei aukati i nga tauhohenga kore. Ko te aroaro o Aib (a-aminoisobutyric acid) e whakatairanga ana i nga hanganga helical me te whakanui i te pumau o te peptide. He mea nui tenei peptide mo te tirotiro i te whakakopa peptide, te whakapumautanga, me te waahi mo te hoahoa peptides hohe koiora.
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BPC-157
Ko te BPC-157 API e whakamahi ana i te tukanga whakahiato wahanga totoka (SPPS):
Te parakore teitei: ≥99% (te kitenga HPLC)
He iti te toenga poke, kahore he endotoxin, kahore he parahanga whakarewa taumaha
Te pumau o te puranga, te kaha tukurua, te tautoko i te whakamahinga taumata werohanga
Tautokohia te taumata karamu me te kirokaramu hei whakatutuki i nga hiahia o nga waahanga rereke mai i te R&D ki te ahumahi.
