; Haina Paclitaxel 33069-62-4 Anti-tumor Botanical Medicine for Ovarian Cancer, Breast Cancer wheketere me nga kaihanga |Gentolex
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Paclitaxel 33069-62-4 Anti-tumor Botanical Medicine for Ovarian Cancer, Breast Cancer

Whakaahuatanga Poto:

Ira whakarewa: 213 °C

Ira kohua: 774.66°C (whakatau tata)

Te hurihanga motuhake: D20 -49°(methanol)

Kiato: 1.0352 (whakatau tata)

Ira hiko: 9°C

Nga tikanga rokiroki: 2-8°C

Puka: paura

Te whakarea kawa: 11.90±0.20(Whakaahua)

Tae: Ma


Taipitopito Hua

Tohu Hua

Taipitopito Hua

Ingoa Paclitaxel
nama CAS 33069-62-4
tātai rāpoi ngota C47H51NO14
Te taumaha ngota 853.92
Tau EINECS 608-826-9
Kohuatanga 774.66°C(I Matapaetia)
Kiato 0.200
Te ahua rokiroki Kua hiri ki te maroke, Rokiroki ki roto i te pouaka tio, 2-8°C
Puka Paura
Tae
Te takai Peeke PE + Peeke Aluminium

Nga kupu taurite

Paclitaxel HCL;Paclitaxel(maoriori);Paclitaxelx;N-BENZYL-BETA-PHENYLISOSERINE ESTER;PACLITAXEL, TAXUS BREVIFOLIA;PACLITAXEL, TAXUS SPECIES;PACLITAXOL;PACLITAXEL

Pānga Rongoā

Whakaahuatanga

Ko te Paclitaxel he diterpenoid monomeric i tangohia mai i te kiri o te tipu maori rongoa Taxus.I kitea e te tirotiro Isotope ko te paclitaxel anake e herea ana ki nga microtubules polymerized, karekau i tauhohe ki nga dimer tubulin korepolymerized.Whai muri i te whakakitenga o nga pūtau ki te paclitaxel, he maha nga microtubules ka kohia ki roto i nga ruma.Ko te kohikohinga o enei microtubules ka pokanoa ki nga momo mahi o nga ruma, ina koa ka mutu te wehenga o nga pūtau i roto i te wahanga mitotic me te aukati i te wehenga noa o nga pūtau.Na roto i te rangahau haumanu Ⅱ-Ⅲ, he pai te nuinga o te paclitaxel mo te mate pukupuku ovarian me te mate pukupuku uma, me te whai hua whakaora mo te mate pukupuku pūkahukahu, mate pukupuku colorectal, melanoma, mate pukupuku mahunga me te kaki, lymphoma me te puku roro.

 

Tohutohu

He painga pai ki te maimoatanga o te mate pukupuku ovarian me te platinum me etahi atu mate pukupuku ovarian me te mate pukupuku uma.Ko te mate pukupuku, ko te mate pukupuku gastrointestinal o runga, ko te pukupuku iti me te mate pukupuku pūtau kore-iti he pai te tirohanga.

 

Whakamahinga

Whakamahia te 1: Nga huaota anti-tumor whanui mo te mate pukupuku ovarian, mate pukupuku uma, aha atu.

Whakamahia te 2: nga huaota anti-tumor whanui whanui mo te maimoatanga o te mate pukupuku ovarian, te mate pukupuku uma me etahi atu mate.

Whakamahia te 3: Nga raau taero antitumor.Mo te maimoatanga o te mate pukupuku mate metastatic me te mate pukupuku ovarian metastatic.Nga huaota anti-tumor whanui whanui mo te maimoatanga o te mate pukupuku ovarian, te mate pukupuku uma me etahi atu mate.

Whakamahia te 4: Te raau taero anti-tumor whai hua;ka herea ki te rohe N-terminal o te β-tubulin, te whakatairanga i nga microtubule tino pumau, te aukati i te depolymerization, te aukati i te wehenga pūtau noa me te mahanga i te wahanga G2/M o te huringa pūtau.

Whakamahia te 5: He tarukino anti-microtubule, te aukati i te depolymerization ma te whakatairanga i te polymerization tubulin, te pupuri i te pumau o te tubulin, me te aukati i te mitosis pūtau.

 

 


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